No

1
2
3

7
8
9

10

11

Nama Senyawa
(3R,4R,5S)-5-amino-4-acetamido3-(propylamino)cyclohex-1-ene-1carboxylic acid
(3R,4R,5S)-5-amino-4-acetamido3-propoxycyclohex-1-ene-1carboxylic acid
(3R,4R,5S)-5-amino-3-propoxy-4(2,2,2trifluoroacetamido)cyclohex-1ene-1-carboxylic acid
(3R,4R,5S)-5-amino-4-acetamido3-(3,3,3trifluoropropoxy)cyclohex-1-ene1-carboxylic acid
(3R,4R,5S)-5-amino-3-{[(2R)-1carboxybutan-2-yl]oxy}-4acetamidocyclohex-1-ene-1carboxylic acid
(3R,4R,5S)-5-amino-3-propoxy-4[(2,2,2trifluoroacetyl)amino]cyclohexene
-1-carboxylic acid
(3R,4R,5S)-5-amino-4-acetamido3-(piperidin-1-yl)cyclohex-1-ene1-carboxylic acid
(3R,4R,5S)-5-amino-3-(azocan-1yl)-4-acetamidocyclohex-1-ene-1carboxylic acid
(3R,4R,5S)-4-acetamido-5-amino3-cyclopentyloxycyclohexene-1carboxylic acid
(3S,4S)-3-carbamimidamido-4[(S)(diethylcarbamoyl)(acetamido)met
hyl]cyclopentane-1-carboxylic
acid
(3S,4S)-3-carbamimidamido-4[(1S)-1-acetamido-2-(morpholin4-yl)-2-oxoethyl]cyclopentane-1carboxylic acid

Ki (M) IC50 (M)

63,77

200

29,32

130

203,37

94,29

262,11

37,49

2,113

2,308

1,974

2,352

2,418

2,653

1,573

0,720

1,397

0,727

1,414

0,675

1,342

0,531

1,176

0,936

1,602

225

450

100

25

5,34

26

4,74

22

8,64

1,467

100

5,25

3,4

1,804

Log
IC50
2,301

Log Ki

15

40