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2. Phenylpiperidine derivates
-fentanyl
-sufentanyl
-alfentanyl
-trimeperidine
3.Benzomorphan derivates
-pantazocine
5. Cyclohexanoles derivates
-thramadol
4. Derivates of cyclohexen-carbonic
acid: -thilidine
6. Morphinane derivates
-butorphanol
7. Opioid antagonist
-naloxone
-nalorphine
-nalmephene
-naltrexone
Non-opioid drugs
1. The salicylates
- acetylsalicylic acid
- sodium salicylate
- methylsalicylate
- salicylamid
2. Pirazolone derivates
-fenylbutazone
-baralgine
II Classification of analgesics
1) With central action:
1. opioid drugs and their antagonists
A)agonist of opioid receptors
a) alkaloids from Papaver somniferum
b). Synthetic drugs
- morphine
- fentanyl
- omnopon
- alfentanyl
- sufentanyl
- thalamonal
- promedol
B)agonist-antagonist and partial agonist of opioid receptors
- pentazocine
- nalbuphine
- butorphanol
C) Antagonists of opioid drugs
-naloxone
-nalorphine
-nalmephene
-naltrexone
Classification of hypnotics
1. Agonist of benzodiazepine receptors.
1) Benzodiazepine derivates
a) Short action T 0,5 1,5-3 hours
- Tiazolam
- Midazolam
- Estazolam
- Ketazolam
b) Medium action T0,5 12-24 hours
- Temazepam
- Nitrazepam
- Lorazepam
- Oxazepam
- Clonazepam
c) Long action T 0,5 30-40 hours
I..Benzodiazepines
- Diazepam
- Flurazepam
- Flunitrazepam
- Fenazepam
II Not benzodiazepines
- Zopiclon
- Zolpidem
- buspiron
II. Hypnotics with anesthetic action (narcotic)
Heterocycles
barbiturics
Medium action
- Pentobarbital
Long action
- Phenobarbital
Aliphatic drugs
- Chloral hydrate
III. Remedies from various groups
- Sedatives
- Tranquilisators
- Neuroleptics (a little doses)
- Antihistamines
**Flumazenil is antagonist of hypnotic drugs
Anti-epileptics
I Partial convulsions
1.psychomotor crisis
- carbamazepine
- phenytoin
- hexamidine
- valproic acid
- phenobarbital
- lamotridgine
- clobazepam
II Generalized convulsions
1) Petit mal (minor crisis)
- ethosuximide
- lamotridgine
- valproic acid
- clonazepam
- thrimetadione
2) Grand mal (major crisis) ( tonic-clonic convulsions)
- phenobarbital
- phenytoin
- valproic acid
- carbamazepine
- lamotridgine
- hexamidine
3) Status epilepticus
- diazepam
- phenobarbital
- lorazepam
- general anesthetics (intravenous)
- clonazepam
4) Myoclonic syndromes
1. valproic acid
2. clonazepam
3. diazepam
4. nitrazepam
5.
III Contractures
a) GABA derivates
b) non benzodiazepines
c) benzodiazepines
Phenibut
tolperyzone
diazepam
baclofen
mefedol
fenazepam
Antiepileptics
Classification 2
I order the drugs administrated in monotherapy
Phenobarbital
Phenytoin
Trimetadione
Ethsuximide
Primidone
Clonazepam
Carbamazepine
Nitrazepam
Valproic acid
Lamotridgine
II order these drugs are associated with I order drugs
Diazepam
Bromides
Acetazolamides
Antiparkinsonian Drugs
1.Remedies that activated dopaminergic system
1) predecessors of dopamine
Levodopa (L Dopa)
Levodopa adjunct (mixed drugs)
- Sinement
- Nacom
- Madopar
- Entancapone
2) dopaminimimetics
- Bromocriptine
3) MAO inhibitor
- Selegeline
2. Remedies that inhibits glutamatergic system
- Amantadine
3. Remedies that inhibits cholinergic system
- Trihexyphenidyl
- Difenyltropine
- Benztropine mesilate
- Triperidine
Psychopharmacologicals
Psychotropic drugs the drugs with the action on the CNS
Classification of Psychotropic drugs
1) Psycholeptics ( inhibit CNS)
- Neuroleptics
- Sedatives
- Tranquilisators
- Lithium
2) Psychoanaleptics (activate CNS)
- Antidepressants
- Nootropes
- Psychostimulants
- Tonisants
- Adaptogenes
3) Psychodyslepics Psychosomimetics
Neuroleptics (antipsychotics)
Typical antipsychotics ( Cause unwanted motor side-effects)
A. Phenothiazines - chlorpromazine
- levomepromazine
- Fluphenazine
- perphenazine
B. Butyrophenones - haloperidol
- trifluperidol
- droperidol
C. Thioxanthenes
- chlothixen
- thiothixene
D. Dyphenylbutylpiperidines
- Fluspirilen
- pimozid
- fenfluridol
Atypical antipsychotics
A Dybenzodiazepines
- clozapin
B Benzamides
- sulpiride
C Alkaloids of Rauwolfia
- rezerpine
Tranquilisators
I .. Major
A Benzodiazepines:
-
Diazepam
Fenazepam
Oxazepam
Nitrazepam
benzoclidine
trimetozine
lonetyl
amixid
librax
antares 120
alrazolam
opipramol
B. Non benzodiazepines
II Minor
proroxane
fenybut
propranolol
mebicar
meprobamat
pyracetam
C Compound drugs
D. Antidepressants
Sedatives drugs
Drugs used to inhibit agitation, stress, and insomnia
Classification:
1) Natural drugs: T-rae Valerian
T-rae Leonur
2) Synthetics
Bromides (Na, K)
3) Barbiturates
Phenobarbital, pentobarbital
4) Compound
Corvalol
Antidepressants
According to the mechanism of action :
A. Amine reuptake blocking drugs
a. nonselective: imipramine, amitriptyline, clomipramine
b. selective:
1) selective serotonine reuptake inhibitors
fluoxetine,
paroxetine
sertraline
2) selective noradrenaline reuptake inhibitors
maprotiline
desipramine
B. Monoamine oxidase inhibitors
a. unreversible drugs
phenelzine
tranylcypromide
nialamide
b. reversible drugs
moclobemide
pirlindol
C. The drugs from various groups with undefined mechanism of action
alprasolam
mianserin
feprozidine
Nootropes
1.
2.
3.
4.
5.
Analeptics
1. Medullar stimulants
- Strychnine,Securenine
2. Bulbs stimulants
- Bemegrid, Niketamine, Pentetrazol
- Camphor, Sulphocomphocaine, Ethimizol
3. General tonizants and adaptogenes
A. Vegetal tonizants: Schizandra, Streculia, Lecozeea,
Echinopanax, Panttocrina, Rantarina
B.Vegetal adaptogens: Panax (Ginseng), Bioginseng,
Eleuterococcus, Rodiola